iphepha_ibhena

iimveliso

I-CAS 23076-35-9 i-hydrochloride

inkcazelo emfutshane:


  • Whatsapp:+8613164690256
  • Wickr:smithliya
  • ITelegram:+8613164690256
  • I-Skype:nguSmith
  • I-imeyile: liya@wh-xiju.com
  • Iinkcukacha zeMveliso

    Iithegi zeMveliso

    5449-12-7

    Igama eliqhelekileyo Xylazine hydrochloride
    Inombolo yeCAS 23076-35-9 Ubunzima beMolekyuli 256.795
    Ukuxinana 1.15g/cm3 Indawo yokubilisa 334.2ºC ku-760mmHg
    Ifomula yeemolekyuli C12H17ClN2S Indawo yokunyibilika 150-164?C (Disemba)
    I-MSDS jgh

    i-USA

    Indawo yokuflasha 155.9ºC
    Uphawu GHS06
    GHS06
    Igama loMqondiso Ingozi

    I-KHJG (3) I-KHJG (4) I-KHJG (1) ukupakisha (6) ukupakisha (7)

    Ukusetyenziswa kwe-Xylazine hydrochloride

    I-Xylazine Hydrochloride yiklasi ye-α2 ye-adrenergic receptor agonist.Ithagethi: I-Adrenergic ReceptorXylazine iyisiyobisi esisetyenziselwa ukutshatyalaliswa, i-anesthesia, ukuphumla kwemisipha, kunye ne-analgesia kwizilwanyana ezifana namahashe, iinkomo kunye nezinye izilwanyana ezingezona abantu.I-analogue ye-clonidine, i-agonist kwiklasi ye-α2 ye-adrenergic receptor.I-Xylazine isanda kuvela njengeyeza lokuzonwabisa, ngakumbi ePuerto Rico [1].Ukulawulwa kwe-xylazine (i-0.17 mg / kg yesisindo somzimba, ihlanjululwe kumthamo we-10-ml, usebenzisa i-0.9% ye-NaCl) yenza malunga neeyure ze-2.5 ze-analgesia yendawo ngaphandle kwemiphumo ebonakalayo.Amanani aphezulu e-xylazine abangela i-ataxia yomlenze ongasemva.Ukulawulwa kwe-lidocaine kubangele ixesha elifanayo le-analgesia, kunye ne-ataxia yangemva enzima (i-100% izehlo).Siye sagqiba kwelokuba i-xylazine enikwe ngenaliti ye-epidural iphumela ekukhuselekeni, okusebenzayo kwe-perineal analgesia kumahashe [2].

    Xylazine hydrochloride Biological Activity

    Inkcazo I-Xylazine Hydrochloride yiklasi ye-α2 ye-adrenergic receptor agonist.Ithagethi: I-Adrenergic ReceptorXylazine iyisiyobisi esisetyenziselwa ukutshatyalaliswa, i-anesthesia, ukuphumla kwemisipha, kunye ne-analgesia kwizilwanyana ezifana namahashe, iinkomo kunye nezinye izilwanyana ezingezona abantu.I-analogue ye-clonidine, i-agonist kwiklasi ye-α2 ye-adrenergic receptor.I-Xylazine isanda kuvela njengeyeza lokuzonwabisa, ngakumbi ePuerto Rico [1].Ukulawulwa kwe-xylazine (i-0.17 mg / kg yesisindo somzimba, ihlanjululwe kumthamo we-10-ml, usebenzisa i-0.9% ye-NaCl) yenza malunga neeyure ze-2.5 ze-analgesia yendawo ngaphandle kwemiphumo ebonakalayo.Amanani aphezulu e-xylazine abangela i-ataxia yomlenze ongasemva.Ukulawulwa kwe-lidocaine kubangele ixesha elifanayo le-analgesia, kunye ne-ataxia yangemva enzima (i-100% izehlo).Siye sagqiba kwelokuba i-xylazine enikwe ngenaliti ye-epidural iphumela ekukhuselekeni, okusebenzayo kwe-perineal analgesia kumahashe [2].
    Ikhathalogu enxulumeneyo
    Iindlela zoMqondiso >> GPCR/G Protein >> I-Adrenergic Receptor
    Iindawo zoPhando >> Izifo zeNeurological
    Isinyibilikisi
    I-In vitro:

    10 mM kwi-DMSO

    Ukunyibilika
    1 mM 3.8942 mL 19.4712 mL 38.9423 mL
    5 mM 0.7788 mL 3.8942 mL 7.7885 ml
    10 mM 0.3894 mL 1.9471 mL 3.8942 mL
    Ugcino
    Umgubo -20°C Iminyaka emi-3
    4°C iminyaka eyi-2
    Kwi-solvent -80°C Iinyanga ezi-6
    -20°C Inyanga eyi-1
    Ukuhambisa ngenqanawe Ubushushu begumbi kwilizwekazi lase-US;zinokwahluka kwenye indawo
    UNCUMILE CC1=C(C(C)=CC=C1)NC2=NCCCS2.Cl
    Iimbekiselo [1].Reyes, JC, et al., Ukuvela kwe-xylazine njengesiyobisi esitsha sokusetyenziswa kakubi kunye nemiphumo yempilo phakathi kwabasebenzisi beziyobisi ePuerto Rico.J Urban Health, 2012. 89(3): p.519-26 [2].I-Hsu, i-WH, i-Xylazine-induced depression kunye ne-antagonism yayo yi-alpha adrenergic blocking agents.J Pharmacol Exp Ther, 1981. 218(1): iphe.188-92.
    Iimolekyuli ezinxulumeneyo Isoprenaline hydrochloride |I-ICI 118,551 (i-hydrochloride) |Phenylephrine hydrochloride |Yohimbine hydrochloride |L(-)-Epinephrine |Ivabradine hydrochloride |Prazosin hydrochloride |Clenbuterol hydrochloride |Phentolamine mesilate |guanfacine hydrochloride |ipimozide |Sotalol hydrochloride |Carvedilol |Atenolol |Metroprolol succinate

    Izithethantonye

    I-BAY 1470 hydrochloride
    Xylazine chloride
    I-2-(2,6-Dimethylphenylamino) -5,6-dihydro-4H-thiazine hydrochloride
    2 - [(2,6-Dimethylphenyl) amino] -5,6-dihydro-4H-1,3-thiazine Hydrochloride
    I-N-(2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine hydrochloride (1: 1)
    BAY VA 1470
    I-EINECS 245-417-0
    I-4H-1,3-Thiazin-2-amine, N-(2,6-dimethylphenyl) -5,6-dihydro-, i-hydrochloride (1: 1)
    I-Celactal
    N-(2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine hydrochloride
    Xylazine HCl
    MFCD00058196

    Inkampani yethu

    I-Wuhan Xiju Biotechnology Co., Ltd. ngumvelisi oqeqeshiweyo wenkqubo ephakathi yamayeza.Inkampani inophando oluzimeleyo kunye neqela lophuhliso, elinokuthi liphande kwaye liphuhlise naziphi na izinto eziluhlaza zonyango, ngexabiso eliphantsi, umgangatho ophezulu kunye nenkonzo yeklasi yokuqala!

    umzimveliso (1) umzi-mveliso (2) umzi-mveliso (3) umzimveliso (4)

    Kutheni Khetha Thina

    I-1, Siqinisekisa uhlalutyo olunzulu kunye nokubonakaliswa, ukucoceka ngaphezu kwe-99.8%.
    2, Umzi-mveliso onexabiso elinomtsalane kunye nesitokhwe esikhulu.
    I-3, indlela yokuhambisa ekhuselekileyo neyingqondi.
    I-4, Sithembisa ukubuyisela imigaqo-nkqubo ukuba isithuba asiphumelelanga okanye ukubuyisela imali xa ufuna.
    I-5, i-Customs clearance rate yi-100% kuquka iRashiya, i-Australia, kunye namanye amazwe.
    6, TNT/UPS/DHL/EMS/FedEx okanye umgca okhethekileyo uyafumaneka kuwe.
    7, Imiqathango yentlawulo: Western Union, Moneygram, Bitcoin, Bank wire ukhetho lwakho.


  • Ngaphambili:
  • Okulandelayo:

  • Bhala umyalezo wakho apha kwaye uwuthumele kuthi