I-CAS 23076-35-9 i-hydrochloride
Igama eliqhelekileyo | Xylazine hydrochloride | ||
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Inombolo yeCAS | 23076-35-9 | Ubunzima beMolekyuli | 256.795 |
Ukuxinana | 1.15g/cm3 | Indawo yokubilisa | 334.2ºC ku-760mmHg |
Ifomula yeemolekyuli | C12H17ClN2S | Indawo yokunyibilika | 150-164?C (Disemba) |
I-MSDS | ![]() | Indawo yokuflasha | 155.9ºC |
Uphawu | ![]() GHS06 | Igama loMqondiso | Ingozi |
Ukusetyenziswa kwe-Xylazine hydrochloride
I-Xylazine Hydrochloride yiklasi ye-α2 ye-adrenergic receptor agonist.Ithagethi: I-Adrenergic ReceptorXylazine iyisiyobisi esisetyenziselwa ukutshatyalaliswa, i-anesthesia, ukuphumla kwemisipha, kunye ne-analgesia kwizilwanyana ezifana namahashe, iinkomo kunye nezinye izilwanyana ezingezona abantu.I-analogue ye-clonidine, i-agonist kwiklasi ye-α2 ye-adrenergic receptor.I-Xylazine isanda kuvela njengeyeza lokuzonwabisa, ngakumbi ePuerto Rico [1].Ukulawulwa kwe-xylazine (i-0.17 mg / kg yesisindo somzimba, ihlanjululwe kumthamo we-10-ml, usebenzisa i-0.9% ye-NaCl) yenza malunga neeyure ze-2.5 ze-analgesia yendawo ngaphandle kwemiphumo ebonakalayo.Amanani aphezulu e-xylazine abangela i-ataxia yomlenze ongasemva.Ukulawulwa kwe-lidocaine kubangele ixesha elifanayo le-analgesia, kunye ne-ataxia yangemva enzima (i-100% izehlo).Siye sagqiba kwelokuba i-xylazine enikwe ngenaliti ye-epidural iphumela ekukhuselekeni, okusebenzayo kwe-perineal analgesia kumahashe [2].
Xylazine hydrochloride Biological Activity
Inkcazo | I-Xylazine Hydrochloride yiklasi ye-α2 ye-adrenergic receptor agonist.Ithagethi: I-Adrenergic ReceptorXylazine iyisiyobisi esisetyenziselwa ukutshatyalaliswa, i-anesthesia, ukuphumla kwemisipha, kunye ne-analgesia kwizilwanyana ezifana namahashe, iinkomo kunye nezinye izilwanyana ezingezona abantu.I-analogue ye-clonidine, i-agonist kwiklasi ye-α2 ye-adrenergic receptor.I-Xylazine isanda kuvela njengeyeza lokuzonwabisa, ngakumbi ePuerto Rico [1].Ukulawulwa kwe-xylazine (i-0.17 mg / kg yesisindo somzimba, ihlanjululwe kumthamo we-10-ml, usebenzisa i-0.9% ye-NaCl) yenza malunga neeyure ze-2.5 ze-analgesia yendawo ngaphandle kwemiphumo ebonakalayo.Amanani aphezulu e-xylazine abangela i-ataxia yomlenze ongasemva.Ukulawulwa kwe-lidocaine kubangele ixesha elifanayo le-analgesia, kunye ne-ataxia yangemva enzima (i-100% izehlo).Siye sagqiba kwelokuba i-xylazine enikwe ngenaliti ye-epidural iphumela ekukhuselekeni, okusebenzayo kwe-perineal analgesia kumahashe [2]. | ||||||||||||
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Ikhathalogu enxulumeneyo | Iindlela zoMqondiso >> GPCR/G Protein >> I-Adrenergic Receptor Iindawo zoPhando >> Izifo zeNeurological | ||||||||||||
Isinyibilikisi | I-In vitro: 10 mM kwi-DMSO | ||||||||||||
Ukunyibilika |
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Ugcino |
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Ukuhambisa ngenqanawe | Ubushushu begumbi kwilizwekazi lase-US;zinokwahluka kwenye indawo | ||||||||||||
UNCUMILE | CC1=C(C(C)=CC=C1)NC2=NCCCS2.Cl | ||||||||||||
Iimbekiselo | [1].Reyes, JC, et al., Ukuvela kwe-xylazine njengesiyobisi esitsha sokusetyenziswa kakubi kunye nemiphumo yempilo phakathi kwabasebenzisi beziyobisi ePuerto Rico.J Urban Health, 2012. 89(3): p.519-26 [2].I-Hsu, i-WH, i-Xylazine-induced depression kunye ne-antagonism yayo yi-alpha adrenergic blocking agents.J Pharmacol Exp Ther, 1981. 218(1): iphe.188-92. | ||||||||||||
Iimolekyuli ezinxulumeneyo | Isoprenaline hydrochloride |I-ICI 118,551 (i-hydrochloride) |Phenylephrine hydrochloride |Yohimbine hydrochloride |L(-)-Epinephrine |Ivabradine hydrochloride |Prazosin hydrochloride |Clenbuterol hydrochloride |Phentolamine mesilate |guanfacine hydrochloride |ipimozide |Sotalol hydrochloride |Carvedilol |Atenolol |Metroprolol succinate |
Izithethantonye
I-BAY 1470 hydrochloride |
Xylazine chloride |
I-2-(2,6-Dimethylphenylamino) -5,6-dihydro-4H-thiazine hydrochloride |
2 - [(2,6-Dimethylphenyl) amino] -5,6-dihydro-4H-1,3-thiazine Hydrochloride |
I-N-(2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine hydrochloride (1: 1) |
BAY VA 1470 |
I-EINECS 245-417-0 |
I-4H-1,3-Thiazin-2-amine, N-(2,6-dimethylphenyl) -5,6-dihydro-, i-hydrochloride (1: 1) |
I-Celactal |
N-(2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine hydrochloride |
Xylazine HCl |
MFCD00058196 |
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